الفهرس 
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Abstract
The reaction of 2-phenyl benzoxazine with p-amino phenol and
ethanol amine lead to formation of quinazolinones 2, 7 that used as chiral
auxiliaries. The reaction of these quinazolinones with different carboxylic
acid derivatives lead to formation of quinazolinone esters 3,8 which
deprotonated with LCHIPA at very low different temperatures followed by
alkylation with different alkyl halide to give quinazolinone α-alkylated
esters 4, 9. The hydrolysis of these esters lead to formation of α- alkylated
acids 5, 10 with high enantiomeric purity.